Drug class · Endocrine & metabolism
DPP-4 inhibitors
Oral drugs that inhibit the dipeptidyl peptidase-4 enzyme, alone or in fixed combinations.
Most-listed names in this class
Ranked by the number of FDA listings, which reflects labelers and package variety — not sales or prescribing.
FDA-listed products
| Product | Strength | Form · route | Labeler | Product NDC |
|---|---|---|---|---|
| Alogliptin | Alogliptin benzoate 25 mg/1 | Tablet, Film coatedOral | Bryant Ranch Prepack | 63629-4946 |
| Alogliptin | Alogliptin benzoate 25 mg/1 | Tablet, Film coatedOral | A-S Medication Solutions | 50090-5574 |
| Alogliptin | Alogliptin benzoate 6.25 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-087 |
| Alogliptin | Alogliptin benzoate 12.5 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-103 |
| Alogliptin | Alogliptin benzoate 12.5 mg/1 | Tablet, Film coatedOral | Aphena Pharma Solutions - Tennessee, LLC | 71610-661 |
| Alogliptin | Alogliptin benzoate 25 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-150 |
| Alogliptin | Alogliptin benzoate 25 mg/1 | Tablet, Film coatedOral | Aphena Pharma Solutions - Tennessee, LLC | 71610-300 |
| Alogliptin and Pioglitazonealogliptin benzoate and pioglitazone hydrochloride | Alogliptin benzoate 12.5 mg/1; Pioglitazone hydrochloride 30 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-260 |
| Alogliptin and Pioglitazonealogliptin benzoate and pioglitazone hydrochloride | Alogliptin benzoate 25 mg/1; Pioglitazone hydrochloride 15 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-351 |
| Alogliptin and Pioglitazonealogliptin benzoate and pioglitazone hydrochloride | Alogliptin benzoate 25 mg/1; Pioglitazone hydrochloride 30 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-402 |
| Alogliptin and Pioglitazonealogliptin benzoate and pioglitazone hydrochloride | Alogliptin benzoate 25 mg/1; Pioglitazone hydrochloride 45 mg/1 | Tablet, Film coatedOral | Padagis Israel Pharmaceuticals Ltd | 45802-499 |
| Brynovinsitagliptin hydrochloride oral | Sitagliptin 25 mg/mL | SolutionOral | Azurity Pharmaceuticals, Inc. | 24338-017 |
| Glyxambiempagliflozin and linagliptin | Empagliflozin 25 mg/1; Linagliptin 5 mg/1 | Tablet, Film coatedOral | Boehringer Ingelheim Pharmaceuticals, Inc. | 0597-0164 |
| Glyxambiempagliflozin and linagliptin | Empagliflozin 10 mg/1; Linagliptin 5 mg/1 | Tablet, Film coatedOral | Boehringer Ingelheim Pharmaceuticals, Inc. | 0597-0182 |
| Janumetsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 1000 mg/1 | Tablet, Film coatedOral | A-S Medication Solutions | 50090-5502 |
| Janumetsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 1000 mg/1 | Tablet, Film coatedOral | Merck Sharp & Dohme LLC | 0006-0577 |
| Janumetsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 500 mg/1 | Tablet, Film coatedOral | A-S Medication Solutions | 50090-5616 |
| Janumetsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 500 mg/1 | Tablet, Film coatedOral | Merck Sharp & Dohme LLC | 0006-0575 |
| Janumet XRsitagliptin and metformin hydrochloride | Sitagliptin phosphate 100 mg/1; Metformin hydrochloride 1000 mg/1 | Tablet, Film coated, Extended releaseOral | Merck Sharp & Dohme LLC | 0006-0081 |
| Janumet XRsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 1000 mg/1 | Tablet, Film coated, Extended releaseOral | A-S Medication Solutions | 50090-5504 |
| Janumet XRsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 500 mg/1 | Tablet, Film coated, Extended releaseOral | Merck Sharp & Dohme LLC | 0006-0078 |
| Janumet XRsitagliptin and metformin hydrochloride | Sitagliptin phosphate 50 mg/1; Metformin hydrochloride 1000 mg/1 | Tablet, Film coated, Extended releaseOral | Merck Sharp & Dohme LLC | 0006-0080 |
| Januviasitagliptin | Sitagliptin phosphate 100 mg/1 | Tablet, Film coatedOral | Merck Sharp & Dohme LLC | 0006-0277 |
| Januviasitagliptin | Sitagliptin phosphate 50 mg/1 | Tablet, Film coatedOral | A-S Medication Solutions | 50090-3472 |
| Januviasitagliptin | Sitagliptin phosphate 100 mg/1 | Tablet, Film coatedOral | A-S Medication Solutions | 50090-1036 |